Date of Award

2015-01-01

Degree Name

Doctor of Philosophy

Department

Chemistry

Advisor(s)

Shizue Mito

Abstract

The total synthesis of Syringolides is described. The synthetic pathway was designed in order to synthesize Syringolides in high yields using inexpensive starting materials. The synthesis strategy features a preparation of the linear tricarbonyl compound followed by intramolecular cyclization. The linear precursor is divided into two fragments, β-keto acid and protected D-xylulose, which are the key fragments and were synthesized from α,β-unsaturated compound followed by asymmetric dihydroxylation. The α,β-unsaturated compound was efficiently prepared by a Wittig reaction between aldehyde and ylide fragments. The butenolide derivative was also achieved by the Knoevenagel condensation of the tricarbonyl compound.

Language

en

Provenance

Received from ProQuest

File Size

84 pages

File Format

application/pdf

Rights Holder

Sudhakar Kalagara

Included in

Chemistry Commons

Share

COinS